Table 3.
Summary of cytostatic activities on seven tumor cell lines presented as median antiproliferative IC50 values and derivatives with IC50 value within the given range.
| A549 |
CFPAC-1 |
SW620 |
HCT-116 |
HeLa |
HepG2 |
MCF-7 |
|
|---|---|---|---|---|---|---|---|
| 8a−8u | |||||||
| Median IC50 | 28.9 | 58.2 | 54.2 | 31.8 | 25.0 | 29.2 | 25.9 |
| IC50 ≥ 100 | 4 | 5 | 7 | 5 | 3 | 3 | 4 |
| IC50 < 30 | 12 | 3 | 3 | 9 | 13 | 11 | 13 |
| IC50 < 1 |
1 |
0 |
0 |
0 |
0 |
0 |
2 |
|
10c−10p |
|||||||
| Median IC50 | 100.0 | 100.0 | 95.8 | 99.4 | 75.8 | 100.0 | 64.6 |
| IC50 ≥ 100 | 11 | 109 | 7 | 7 | 6 | 8 | 6 |
| IC50 < 30 | 2 | 0 | 3 | 1 | 4 | 0 | 4 |
| IC50 < 1 | 0 | 0 | 0 | 0 | 0 | 0 | 0 |