Table 4.
Enzyme and cellular activities of amides S27, S28 and S29.
| Com. | IC50 MetAP2 (nM) | GI50 HUVEC (μM) | GI @ 5 μM HUVEC (%) |
|---|---|---|---|
| S27 | 177 | 0.67 | >98 |
| S28 | 755 | – | 93 |
| S29 | 67 | 0.85 | >98 |
Official websites use .gov
A
.gov website belongs to an official
government organization in the United States.
Secure .gov websites use HTTPS
A lock (
) or https:// means you've safely
connected to the .gov website. Share sensitive
information only on official, secure websites.