Table 1.
Receptor parameters
| Parameter | Source | |
|---|---|---|
| Measured values | ||
| [D1]m in pmol/mg protein | 2.840 | Richfield et al. (1989a) |
| [D2]m in pmol/mg protein | 0.696 | Richfield et al. (1989a) |
| ϵ | 0.12 | Banay-Schwartz et al. (1992) |
| α | 0.2 | Syková and Nicholson (2008) |
| ρbrain in g/ml | 1.05 | DiResta et al. (1990) |
| fD1membrane | 1.0 | Prou et al. (2001) |
| fD2membrane | 0.2 | Prou et al. (2001) |
| konD1,orig in nM−1 min−1 | 0.00025 | Sano et al. (1979) |
| koffD1,orig in min−1 | 0.64 | Sano et al. (1979) |
| konD2 in nM−1 min−1 | 0.02 | Burt et al. (1976) |
| koffD2 in min−1 | 0.5 | Burt et al. (1976) |
| [D1]tot in nM | ≈1600 | Equation 17 |
| [D2]tot in nM | ≈80 | Equation 17 |
| konD1,used in nM−1 min−1 | 0.0003125 | see Text |
| koffD1,used in min−1 | 0.5 | see Text |