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. 2020 Apr 1;40(14):2868–2881. doi: 10.1523/JNEUROSCI.1951-19.2019

Table 1.

Receptor parameters

Parameter Source
Measured values
    [D1]m in pmol/mg protein 2.840 Richfield et al. (1989a)
    [D2]m in pmol/mg protein 0.696 Richfield et al. (1989a)
    ϵ 0.12 Banay-Schwartz et al. (1992)
    α 0.2 Syková and Nicholson (2008)
    ρbrain in g/ml 1.05 DiResta et al. (1990)
    fD1membrane 1.0 Prou et al. (2001)
    fD2membrane 0.2 Prou et al. (2001)
    konD1,orig in nM−1 min−1 0.00025 Sano et al. (1979)
    koffD1,orig in min−1 0.64 Sano et al. (1979)
    konD2 in nM−1 min−1 0.02 Burt et al. (1976)
    koffD2 in min−1 0.5 Burt et al. (1976)
    [D1]tot in nM ≈1600 Equation 17
    [D2]tot in nM ≈80 Equation 17
    konD1,used in nM−1 min−1 0.0003125 see Text
    koffD1,used in min−1 0.5 see Text