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. Author manuscript; available in PMC: 2021 Apr 3.
Published in final edited form as: ChemMedChem. 2020 Feb 14;15(7):643–658. doi: 10.1002/cmdc.201900730

Table 3.

Antiproliferative activities of 1–3 on MV4–11 AML and NB4 APL cell lines.

Compd Metabolic stability data[a]
Mouse Clint (μL/min/mg protein) Human Clint (μL/min/mg protein)
3a 7.1 ± 2.2 6.7 ± 1.1
3d 4.3 ± 0.7 12.2 ± 1.7
3g 11.2 ± 1.8 lower than 3
[a]

Data are expressed as the mean of at least two determinations ± standard deviation.