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. 2010 Mar 1;18(7):2439–2446. doi: 10.1016/j.bmc.2010.02.059

Scheme 1.

Scheme 1

Reagents and conditions: (i) DMF, diphenyl carbonate, 100 °C, K2CO3, 137 °C, 1.5 h; (ii) H2O, HCl (2 N), 80 °C, 2 h.