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. 2020 Apr 8;11:408. doi: 10.3389/fphar.2020.00408

Table 1.

Autophagy inhibitors in cancer cells.

Autophagy inhibitor Target point Inhibition stage References
3-MA PI3K inhibition Early (Horwacik et al., 2015; Zhang et al., 2015)
LY294002 PI3K/mTOR inhibition Early (Feng et al., 2018; Shen et al., 2017)
Baf A1 Vacuolar-type H(+)-ATPase inhibition Late (Miyazawa, 2011)
CQ Lysosomal inhibition Late (Kimura et al., 2012; Fukuda et al., 2015; Liu et al., 2016)
HCQ Lysosomal inhibition Late (Vogl et al., 2014; Rangwala et al., 2014)
ABT-737 Bcl-2 inhibition Early (Huang and Sinicrope, 2010; Yang et al., 2016)
Obatoclax Lysosomal inhibition Late (Koehler et al., 2015; Jiménez-Guerrero et al., 2018)
Clarithromycin Block autophagy flux Late (Altman and Platanias, 2012; Sugita et al., 2015)
Resveratrol Autophagy regulator -S6K1 Early (Lin et al., 2012; Alayev et al., 2015; Rai et al., 2016)
Quinacrine Lysosomal inhibition Late (Lobo et al., 2013; Golden et al., 2015)
4-Acetylantroquinonol B Block autophagy flux Late (Liu et al., 2017)
EGCG Block autophagy flux Late (Meng et al., 2019)

3-MA, 3-methyladenine; Baf A1, bafilomycin A1; PI3K, phosphatidylinositol 3 kinase; mTOR, mammalian target of rapamycin; CQ, chloroquine; HCQ, hydroxychloroquine; ATPase, adenosine triphosphatase; EGCG, Epigallocatechin gallate.