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. 2003 Jan 28;68(2):125–132. doi: 10.1016/S0039-128X(02)00166-6

Scheme 1.

Scheme 1

Conditions: (a) p-TsCl, pyridine; (b) LiCO3, LiBr, DMF; (c) m-ClPBA, H2O-CH2Cl2; (d) H2SO4, THF.