Table 2. Fitted slope factor of conductance vs voltage relationship of Kv7.1/KCNE1 + PUFA analogues.
PUFA Analogue | Control | 0.2 mM | 0.7 mM | 2 mM | 7 mM | 20 mM |
---|---|---|---|---|---|---|
Lin-taurine | 17.5 ± 0.75 mV | 17.7 ± 0.76 mV | 17.7 ± 0.77 mV | 18.6 ± 1.0 mV | 18.1 ± 1.0 mV | 12.2 ± 1.8 mV |
N-AT | 16.7 ± 0.71 mV | 16.9 ± 0.65 mV | 17.2 ± 0.62 mV | 17.4 ± 0.60 mV | 18.2 ± 0.59 mV | 18.7 ± 0.73 mV |
Pin-taurine | 17.7 ± 0.67 mV | 17.9 ± 0.82 mV | 17.7 ± 0.82 mV | 18.3 ± 0.96 mV | 18.8 ± 1.0 mV | 16.8 ± 0.73 mV |
DHA-taurine | 18.7 ± 1.2 mV | 18.7 ± 1.1 mV | 18.6 ± 1.2 mV | 18.6 ± 1.3 mV | 18.1 ± 1.2 mV | NA |
Lin-glycine | 18.4 ± 1.2 mV | 18.2 ± 0.89 mV | 19.0 ± 1.0 mV | 19.2 ± 1.2 mV | 20.6 ± 1.5 mV | 22.1 ± 1.7 mV |
Pin-glycine | 18.4 ± 0.70 mV | 17.9 ± 0.83 mV | 17.8 ± 0.84 mV | 17.9 ± 0.91 mV | 18.7 ± 1.1 mV | 20.9 ± 1.4 mV |
DHA-glycine | 16.7 ± 0.44 mV | 16.5 ± 0.49 mV | 16.6 ± 0.45 mV | 16.6 ± 0.52 mV | 17.0 ± 0.56 mV | 17.9 ± 0.68 mV |