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. 2020 Mar 9;50(4):349–356. doi: 10.1093/jjco/hyaa004

Table 3.

Clinical use of PSMA ligands (Oct 2019)

18F-PSMA ligands Organization or company Clinical phase
1 18F-DCFPyL Progenics Pharmaceuticals Phase 3
2 18F-PSMA-1007 ABX Clinical study
3 18F-CTT1057 Novartis (AAA) Phase 1
4 18F-rhPSMA-7.3 Blue Earth Diagnostics Phase 1
5 18F-FSU-880 Kyoto University Phase 2
68 Ga-PSMA ligands Organization or company Clinical phase
1 68Ga-PSMA-11 Telix Pharmaceuticals Phase 3
2 68Ga-PSMA-617 Novartis (Endocyte) Clinical study
3 68Ga-PSMA-I&T Technical University of Munich Clinical study
PSMA ligands for RLT Organization or company Clinical phase
1 177Lu-PSMA-617 Novartis (Endocyte) Phase 3
2 225Ac-PSMA-617 Novartis (Endocyte) Phase 1
3 177Lu-TX591 Telix Pharmaceuticals Phase 2
4 177Lu-PSMA-R2 Novartis (AAA) Phase 1/2
5 227Th-PSMA-TTC Bayer Phase 1

Abbreviation: RLT, radioligand therapy.