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. 2008 Sep 10;275(20):4980–4989. doi: 10.1111/j.1742-4658.2008.06631.x

Table 1.

 Inhibitory characteristics and K i values of diferent tarocystatin segments.

Model Average (%) inhibitory activity K i value (μm)
FL peptide (group‐2) mixed inhibition 55 K ia 0.098, K ib 0.252
Nt peptide (group‐1) competitive inhibition 39 K i 0.057
Ct peptide allosteric activation −18