Table I.
Viral‐Entry Inhibition Activity of Heptad Repeat Peptides and Small Molecules
Peptide | EC50 (µM)a |
---|---|
His6‐HR1 | ND |
GST‐removed HR2 | 2.15 |
HR1‐a | 1.16 |
HR1‐b | ND |
HR2 | 0.34 |
Small molecule | EC50 (µM) |
---|---|
HKC‐5 | 38.38 |
HKC‐21 | 35.94 |
HKC‐24 | 32.60 |
HKC‐25 | 18.74 |
ADS‐J1 | 3.89 |
Quercetin | 64.80 |
XXT | ND |
ND, not detectable.
All measurements were average values of triplicates.