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. 2008 Apr 28;104(6):2335–2347. doi: 10.1002/jcb.21790

Table I.

Viral‐Entry Inhibition Activity of Heptad Repeat Peptides and Small Molecules

Peptide EC50 (µM)a
His6‐HR1 ND
GST‐removed HR2 2.15
HR1‐a 1.16
HR1‐b ND
HR2 0.34
Small molecule EC50 (µM)
HKC‐5 38.38
HKC‐21 35.94
HKC‐24 32.60
HKC‐25 18.74
ADS‐J1 3.89
Quercetin 64.80
XXT ND

ND, not detectable.

a

All measurements were average values of triplicates.