Table 1. Potency distribution for the 4195 HTS primary actives that were progressed to dose-response experiments (Yeast HTS Growth Assay).
pEC50 range | # of Cmpds | % of Cmpds |
---|---|---|
<4 | 3299 | 77% |
4 < × < 4.99 | 741 | 18% |
5 < × < 5.49 | 156 | 3.7% |
5.5 < × < 5.99 | 53 | 1.3% |
6 < × < 6.49 | 13 | 0.3% |
6.5 < × < 6.59 | 2 | 0.05% |