Table 1.
Receptors Identified in Mediating Cannabidiol Immune Effects
Receptor | Activity | References |
---|---|---|
CB1 | Agonist | 58 |
CB2 | Agonist | 59,60 |
FAAH | Inhibition | 58,65–67,84,157,160 |
TRPV1 | Agonist | 65,66,74,82–88,105,148,194 |
Adenosine A2A | Agonist | 89–91,125,164 |
PPAR-γ | Activation | 92–94,96–98,136 |
5-HT1a | Agonist | 59 |
GPR55 | Antagonist | 109,110 |
FAAH, fatty acid amide hydrolase; PPAR-γ, peroxisome proliferator-activated receptor gamma; TRPV1, transient receptor potential vanilloid 1.