Table 1.

IC₅₀ values of selective late sodium current inhibitors for the late and the early sodium current component.

Compound	IC50 for		Reference
	INa,late	INa,early
Lidocaine	29 µM	367 µM	Antzelevitch et al., 2014
Ranolazine	17 µM	1329 µM	Belardinelli et al., 2013
	6 µM	294 µM	Undrovinas et al., 2006
GS-458967	333 nM	<15 % block at 333 nM	Koltun et al., 2016a
	130 nM	7.5 % reduction at 10 µM	Belardinelli et al., 2013
GS-462808	1.9 µM	10 % reduction at 10 µM	Koltun et al., 2016b
GS-6615	0.62 µM	51 µM	Zablocki et al., 2016
F15845	3.25 µM	23 % reduction at 10 µM	Vacher et al., 2009

Where the IC₅₀ value is missing, inhibition percentage at a given concentration was used instead.