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. 2020 Apr 28;40(4):BSR20192920. doi: 10.1042/BSR20192920

Table 3. Information for target genes of tripterygium from TCMSP database.

Mol Id Gene Name Mol name
MOL000296 PGR hederagenin
MOL000296 NCOA2 hederagenin
MOL000296 CHRM3 hederagenin
MOL000296 CHRM1 hederagenin
MOL000296 CHRM2 hederagenin
MOL000296 ADRA1B hederagenin
MOL000296 GABRA1 hederagenin
MOL000296 GRIA2 hederagenin
MOL000296 ADH1B hederagenin
MOL000296 ADH1C hederagenin
MOL000296 LYZ hederagenin
MOL000296 PTGS1 hederagenin
MOL000296 SCN5A hederagenin
MOL000296 PTGS2 hederagenin
MOL000296 RXRA hederagenin
MOL000296 SLC6A2 hederagenin
MOL003182 KCNH2 (+)-Medioresinol di-O-beta-D-glucopyranoside_qt
MOL003182 SCN5A (+)-Medioresinol di-O-beta-D-glucopyranoside_qt
MOL003182 PTGS2 (+)-Medioresinol di-O-beta-D-glucopyranoside_qt
MOL003182 F7 (+)-Medioresinol di-O-beta-D-glucopyranoside_qt
MOL003184 PTGS1 81827-74-9
MOL003184 CHRM3 81827-74-9
MOL003184 KCNH2 81827-74-9
MOL003184 CHRM1 81827-74-9
MOL003184 SCN5A 81827-74-9
MOL003184 CHRM5 81827-74-9
MOL003184 PTGS2 81827-74-9
MOL003184 CHRM4 81827-74-9
MOL003184 OPRD1 81827-74-9
MOL003184 PGR 81827-74-9
MOL003184 CHRM2 81827-74-9
MOL003184 ADRA1B 81827-74-9
MOL003184 ADRB2 81827-74-9
MOL003184 OPRM1 81827-74-9
MOL003184 NCOA2 81827-74-9
MOL003184 NCOA1 81827-74-9
MOL003185 CHRM3 (1R,4aR,10aS)-5-hydroxy-1-(hydroxymethyl)-7-isopropyl-8-methoxy-1,4a
-dimethyl-4,9,10,10a-tetrahydro-3H-phenanthren-2-one
MOL003185 CHRM1 (1R,4aR,10aS)-5-hydroxy-1-(hydroxymethyl)-7-isopropyl-8-methoxy-1,4a-dimethyl
-4,9,10,10a-tetrahydro-3H-phenanthren-2-one
MOL003185 PTGS2 (1R,4aR,10aS)-5-hydroxy-1-(hydroxymethyl)-7-isopropyl-8-methoxy-1,4a-dimethyl
-4,9,10,10a-tetrahydro-3H-phenanthren-2-one
MOL003185 OPRD1 (1R,4aR,10aS)-5-hydroxy-1-(hydroxymethyl)-7-isopropyl-8-methoxy-1,4a-dimethyl
-4,9,10,10a-tetrahydro-3H-phenanthren-2-one
MOL003185 ADRA1A (1R,4aR,10aS)-5-hydroxy-1-(hydroxymethyl)-7-isopropyl-8-methoxy-1,4a-dimethyl-
4,9,10,10a-tetrahydro-3H-phenanthren-2-one
MOL003185 ADRA1B (1R,4aR,10aS)-5-hydroxy-1-(hydroxymethyl)-7-isopropyl-8-methoxy-1,4a-dimethyl-
4,9,10,10a-tetrahydro-3H-phenanthren-2-one
MOL003185 ADRA1D (1R,4aR,10aS)-5-hydroxy-1-(hydroxymethyl)-7-isopropyl-8-methoxy-1,4a-dimethyl-
4,9,10,10a-tetrahydro-3H-phenanthren-2-one
MOL003185 OPRM1 (1R,4aR,10aS)-5-hydroxy-1-(hydroxymethyl)-7-isopropyl-8-methoxy-1,4a-dimethyl-
4,9,10,10a-tetrahydro-3H-phenanthren-2-one
MOL003185 NR3C1 (1R,4aR,10aS)-5-hydroxy-1-(hydroxymethyl)-7-isopropyl-8-methoxy-1,4a-dimethyl-
4,9,10,10a-tetrahydro-3H-phenanthren-2-one
MOL003185 NCOA2 (1R,4aR,10aS)-5-hydroxy-1-(hydroxymethyl)-7-isopropyl-8-methoxy-1,4a-dimethyl-
4,9,10,10a-tetrahydro-3H-phenanthren-2-one
MOL003185 NCOA1 (1R,4aR,10aS)-5-hydroxy-1-(hydroxymethyl)-7-isopropyl-8-methoxy-1,4a-dimethyl-
4,9,10,10a-tetrahydro-3H-phenanthren-2-one
MOL003185 SCN5A (1R,4aR,10aS)-5-hydroxy-1-(hydroxymethyl)-7-isopropyl-8-methoxy-1,4a-dimethyl-
4,9,10,10a-tetrahydro-3H-phenanthren-2-one
MOL003185 CHRM2 (1R,4aR,10aS)-5-hydroxy-1-(hydroxymethyl)-7-isopropyl-8-methoxy-1,4a-dimethyl-
4,9,10,10a-tetrahydro-3H-phenanthren-2-one
MOL003185 ADRB2 (1R,4aR,10aS)-5-hydroxy-1-(hydroxymethyl)-7-isopropyl-8-methoxy-1,4a-dimethyl-
4,9,10,10a-tetrahydro-3H-phenanthren-2-one
MOL003187 RELA triptolide
MOL003187 STAT3 triptolide
MOL003187 VEGFA triptolide
MOL003187 BCL2 triptolide
MOL003187 FOS triptolide
MOL003187 CDKN1A triptolide
MOL003187 PLAU triptolide
MOL003187 TNFSF15 triptolide
MOL003187 JUN triptolide
MOL003187 CASP3 triptolide
MOL003187 TP63 triptolide
MOL003187 MAPK8 triptolide
MOL003187 PTGS2 triptolide
MOL003187 STAT1 triptolide
MOL003187 CXCL8 triptolide
MOL003187 MCL1 triptolide
MOL003187 IL2 triptolide
MOL003187 IFNG triptolide
MOL003187 IL4 triptolide
MOL003187 CD80 triptolide
MOL003187 CD86 triptolide
MOL003187 CXCR4 triptolide
MOL003187 BIRC3 triptolide
MOL003187 CD274 triptolide
MOL003187 IL23A triptolide
MOL003187 CCR7 triptolide
MOL003187 CD1A triptolide
MOL003187 CD40 triptolide
MOL003187 CD14 triptolide
MOL003187 C3 triptolide
MOL003187 VTCN1 triptolide
MOL003196 CHRM3 Tryptophenolide
MOL003196 KCNH2 Tryptophenolide
MOL003196 CHRM1 Tryptophenolide
MOL003196 SCN5A Tryptophenolide
MOL003196 CHRM5 Tryptophenolide
MOL003196 PTGS2 Tryptophenolide
MOL003196 RXRA Tryptophenolide
MOL003196 OPRD1 Tryptophenolide
MOL003196 ADRA1A Tryptophenolide
MOL003196 PGR Tryptophenolide
MOL003196 CHRM2 Tryptophenolide
MOL003196 ADRA1B Tryptophenolide
MOL003196 ADRB2 Tryptophenolide
MOL003196 ADRA1D Tryptophenolide
MOL003196 OPRM1 Tryptophenolide
MOL003196 NCOA2 Tryptophenolide
MOL003196 NCOA1 Tryptophenolide
MOL003199 NOS2 5,8-Dihydroxy-7-(4-hydroxy-5-methyl-coumarin-3)-coumarin
MOL003199 PTGS1 5,8-Dihydroxy-7-(4-hydroxy-5-methyl-coumarin-3)-coumarin
MOL003199 KCNH2 5,8-Dihydroxy-7-(4-hydroxy-5-methyl-coumarin-3)-coumarin
MOL003199 ESR1 5,8-Dihydroxy-7-(4-hydroxy-5-methyl-coumarin-3)-coumarin
MOL003199 AR 5,8-Dihydroxy-7-(4-hydroxy-5-methyl-coumarin-3)-coumarin
MOL003199 SCN5A 5,8-Dihydroxy-7-(4-hydroxy-5-methyl-coumarin-3)-coumarin
MOL003199 PPARG 5,8-Dihydroxy-7-(4-hydroxy-5-methyl-coumarin-3)-coumarin
MOL003199 PTGS2 5,8-Dihydroxy-7-(4-hydroxy-5-methyl-coumarin-3)-coumarin
MOL003199 F7 5,8-Dihydroxy-7-(4-hydroxy-5-methyl-coumarin-3)-coumarin
MOL003199 KDR 5,8-Dihydroxy-7-(4-hydroxy-5-methyl-coumarin-3)-coumarin
MOL003199 PYGM 5,8-Dihydroxy-7-(4-hydroxy-5-methyl-coumarin-3)-coumarin
MOL003199 PRSS1 5,8-Dihydroxy-7-(4-hydroxy-5-methyl-coumarin-3)-coumarin
MOL003209 KCNH2 Celallocinnine
MOL003209 SCN5A Celallocinnine
MOL003217 NOS2 Isoxanthohumol
MOL003217 KCNH2 Isoxanthohumol
MOL003217 ESR1 Isoxanthohumol
MOL003217 SCN5A Isoxanthohumol
MOL003217 PTGS2 Isoxanthohumol
MOL003217 KDR Isoxanthohumol
MOL003217 ADRA1B Isoxanthohumol
MOL003217 ADRB2 Isoxanthohumol
MOL003217 NCOA2 Isoxanthohumol
MOL003217 NCOA1 Isoxanthohumol
MOL003217 PTGS1 Isoxanthohumol
MOL003217 PPARD Isoxanthohumol
MOL003224 NR3C2 Tripdiotolnide
MOL003225 NR3C2 Hypodiolide A
MOL003225 NR3C1 Hypodiolide A
MOL003229 CHRM3 Triptinin B
MOL003229 KCNH2 Triptinin B
MOL003229 CHRM1 Triptinin B
MOL003229 SCN5A Triptinin B
MOL003229 CHRM5 Triptinin B
MOL003229 PTGS2 Triptinin B
MOL003229 RXRA Triptinin B
MOL003229 ADRA1A Triptinin B
MOL003229 PGR Triptinin B
MOL003229 CHRM2 Triptinin B
MOL003229 ADRA1B Triptinin B
MOL003229 ADRB2 Triptinin B
MOL003229 ADRA1D Triptinin B
MOL003229 OPRM1 Triptinin B
MOL003229 NR3C1 Triptinin B
MOL003229 RXRB Triptinin B
MOL003229 NCOA2 Triptinin B
MOL003229 NCOA1 Triptinin B
MOL003231 PTGS1 Triptoditerpenic acid B
MOL003231 CHRM3 Triptoditerpenic acid B
MOL003231 KCNH2 Triptoditerpenic acid B
MOL003231 CHRM1 Triptoditerpenic acid B
MOL003231 SCN5A Triptoditerpenic acid B
MOL003231 CHRM5 Triptoditerpenic acid B
MOL003231 PTGS2 Triptoditerpenic acid B
MOL003231 CHRM4 Triptoditerpenic acid B
MOL003231 RXRA Triptoditerpenic acid B
MOL003231 OPRD1 Triptoditerpenic acid B
MOL003231 ADRA1A Triptoditerpenic acid B
MOL003231 PGR Triptoditerpenic acid B
MOL003231 CHRM2 Triptoditerpenic acid B
MOL003231 ADRA1B Triptoditerpenic acid B
MOL003231 ADRB2 Triptoditerpenic acid B
MOL003231 ADRA1D Triptoditerpenic acid B
MOL003231 OPRM1 Triptoditerpenic acid B
MOL003231 NR3C1 Triptoditerpenic acid B
MOL003231 RXRB Triptoditerpenic acid B
MOL003231 NCOA2 Triptoditerpenic acid B
MOL003231 NCOA1 Triptoditerpenic acid B
MOL003245 CHRM3 Triptonoditerpenic acid
MOL003245 KCNH2 Triptonoditerpenic acid
MOL003245 CHRM1 Triptonoditerpenic acid
MOL003245 SCN5A Triptonoditerpenic acid
MOL003245 PTGS2 Triptonoditerpenic acid
MOL003245 OPRD1 Triptonoditerpenic acid
MOL003245 ADRA1B Triptonoditerpenic acid
MOL003245 ADRB2 Triptonoditerpenic acid
MOL003245 NCOA2 Triptonoditerpenic acid
MOL003245 NCOA1 Triptonoditerpenic acid
MOL003248 PTGS1 Triptonoterpene
MOL003248 CHRM3 Triptonoterpene
MOL003248 CHRM1 Triptonoterpene
MOL003248 SCN5A Triptonoterpene
MOL003248 PTGS2 Triptonoterpene
MOL003248 RXRA Triptonoterpene
MOL003248 ACHE Triptonoterpene
MOL003248 ADRA1A Triptonoterpene
MOL003248 PGR Triptonoterpene
MOL003248 CHRM2 Triptonoterpene
MOL003248 ADRA1B Triptonoterpene
MOL003248 ADRB2 Triptonoterpene
MOL003248 ADRA1D Triptonoterpene
MOL003248 OPRM1 Triptonoterpene
MOL003248 NR3C1 Triptonoterpene
MOL003248 NCOA2 Triptonoterpene
MOL003248 NCOA1 Triptonoterpene
MOL003266 PGR 21-Hydroxy-30-norhopan-22-one
MOL003280 CHRM3 TRIPTONOLIDE
MOL003280 CHRM1 TRIPTONOLIDE
MOL003280 SCN5A TRIPTONOLIDE
MOL003280 CHRM5 TRIPTONOLIDE
MOL003280 PTGS2 TRIPTONOLIDE
MOL003280 OPRD1 TRIPTONOLIDE
MOL003280 ADRA1A TRIPTONOLIDE
MOL003280 PGR TRIPTONOLIDE
MOL003280 CHRM2 TRIPTONOLIDE
MOL003280 ADRB2 TRIPTONOLIDE
MOL003280 OPRM1 TRIPTONOLIDE
MOL003280 NCOA2 TRIPTONOLIDE
MOL003280 NCOA1 TRIPTONOLIDE
MOL000358 PGR beta-sitosterol
MOL000358 NCOA2 beta-sitosterol
MOL000358 PTGS1 beta-sitosterol
MOL000358 PTGS2 beta-sitosterol
MOL000358 KCNH2 beta-sitosterol
MOL000358 CHRM3 beta-sitosterol
MOL000358 CHRM1 beta-sitosterol
MOL000358 SCN5A beta-sitosterol
MOL000358 CHRM4 beta-sitosterol
MOL000358 ADRA1A beta-sitosterol
MOL000358 CHRM2 beta-sitosterol
MOL000358 ADRA1B beta-sitosterol
MOL000358 ADRB2 beta-sitosterol
MOL000358 CHRNA2 beta-sitosterol
MOL000358 SLC6A4 beta-sitosterol
MOL000358 OPRM1 beta-sitosterol
MOL000358 GABRA1 beta-sitosterol
MOL000358 BCL2 beta-sitosterol
MOL000358 BAX beta-sitosterol
MOL000358 CASP9 beta-sitosterol
MOL000358 JUN beta-sitosterol
MOL000358 CASP3 beta-sitosterol
MOL000358 CASP8 beta-sitosterol
MOL000358 PRKCA beta-sitosterol
MOL000358 PON1 beta-sitosterol
MOL000358 MAP2 beta-sitosterol
MOL000211 PGR Mairin
MOL000422 NOS2 kaempferol
MOL000422 PTGS1 kaempferol
MOL000422 AR kaempferol
MOL000422 PPARG kaempferol
MOL000422 PTGS2 kaempferol
MOL000422 NCOA2 kaempferol
MOL000422 PRSS1 kaempferol
MOL000422 PGR kaempferol
MOL000422 CHRM1 kaempferol
MOL000422 ACHE kaempferol
MOL000422 SLC6A2 kaempferol
MOL000422 CHRM2 kaempferol
MOL000422 ADRA1B kaempferol
MOL000422 GABRA1 kaempferol
MOL000422 F7 kaempferol
MOL000422 RELA kaempferol
MOL000422 IKBKB kaempferol
MOL000422 AKT1 kaempferol
MOL000422 BCL2 kaempferol
MOL000422 BAX kaempferol
MOL000422 TNFSF15 kaempferol
MOL000422 JUN kaempferol
MOL000422 AHSA1 kaempferol
MOL000422 CASP3 kaempferol
MOL000422 MAPK8 kaempferol
MOL000422 MMP1 kaempferol
MOL000422 STAT1 kaempferol
MOL000422 PPARG kaempferol
MOL000422 HMOX1 kaempferol
MOL000422 CYP3A4 kaempferol
MOL000422 CYP1A2 kaempferol
MOL000422 CYP1A1 kaempferol
MOL000422 ICAM1 kaempferol
MOL000422 SELE kaempferol
MOL000422 VCAM1 kaempferol
MOL000422 NR1I2 kaempferol
MOL000422 CYP1B1 kaempferol
MOL000422 ALOX5 kaempferol
MOL000422 HAS2 kaempferol
MOL000422 GSTP1 kaempferol
MOL000422 AHR kaempferol
MOL000422 PSMD3 kaempferol
MOL000422 SLC2A4 kaempferol
MOL000422 NR1I3 kaempferol
MOL000422 INSR kaempferol
MOL000422 DIO1 kaempferol
MOL000422 PPP3CA kaempferol
MOL000422 GSTM1 kaempferol
MOL000422 GSTM2 kaempferol
MOL000422 AKR1C3 kaempferol
MOL000422 SLPI kaempferol
MOL000449 PGR Stigmasterol
MOL000449 NR3C2 Stigmasterol
MOL000449 NCOA2 Stigmasterol
MOL000449 ADH1C Stigmasterol
MOL000449 RXRA Stigmasterol
MOL000449 NCOA1 Stigmasterol
MOL000449 PTGS1 Stigmasterol
MOL000449 PTGS2 Stigmasterol
MOL000449 ADRA2A Stigmasterol
MOL000449 SLC6A2 Stigmasterol
MOL000449 SLC6A3 Stigmasterol
MOL000449 ADRB2 Stigmasterol
MOL000449 AKR1B1 Stigmasterol
MOL000449 PLAU Stigmasterol
MOL000449 LTA4H Stigmasterol
MOL000449 MAOB Stigmasterol
MOL000449 MAOA Stigmasterol
MOL000449 CTRB1 Stigmasterol
MOL000449 CHRM3 Stigmasterol
MOL000449 CHRM1 Stigmasterol
MOL000449 ADRB1 Stigmasterol
MOL000449 SCN5A Stigmasterol
MOL000449 ADRA1A Stigmasterol
MOL000449 CHRM2 Stigmasterol
MOL000449 ADRA1B Stigmasterol
MOL000449 GABRA1 Stigmasterol
MOL002058 KCNH2 40957-99-1
MOL002058 SCN5A 40957-99-1
MOL002058 PTGS2 40957-99-1
MOL002058 PTGS1 40957-99-1
MOL002058 NCOA2 40957-99-1
MOL002058 F7 40957-99-1
MOL003283 ESR1 (2R,3R,4S)-4-(4-hydroxy-3-methoxy-phenyl)-7-methoxy-2,3-dimethylol-tetralin-6-ol
MOL003283 AR (2R,3R,4S)-4-(4-hydroxy-3-methoxy-phenyl)-7-methoxy-2,3-dimethylol-tetralin-6-ol
MOL003283 PPARG (2R,3R,4S)-4-(4-hydroxy-3-methoxy-phenyl)-7-methoxy-2,3-dimethylol-tetralin-6-ol
MOL003283 PTGS2 (2R,3R,4S)-4-(4-hydroxy-3-methoxy-phenyl)-7-methoxy-2,3-dimethylol-tetralin-6-ol
MOL003283 F7 (2R,3R,4S)-4-(4-hydroxy-3-methoxy-phenyl)-7-methoxy-2,3-dimethylol-tetralin-6-ol
MOL003283 ADRB2 (2R,3R,4S)-4-(4-hydroxy-3-methoxy-phenyl)-7-methoxy-2,3-dimethylol-tetralin-6-ol
MOL003283 ESR2 (2R,3R,4S)-4-(4-hydroxy-3-methoxy-phenyl)-7-methoxy-2,3-dimethylol-tetralin-6-ol
MOL003283 MAPK14 (2R,3R,4S)-4-(4-hydroxy-3-methoxy-phenyl)-7-methoxy-2,3-dimethylol-tetralin-6-ol
MOL003283 GSK3B (2R,3R,4S)-4-(4-hydroxy-3-methoxy-phenyl)-7-methoxy-2,3-dimethylol-tetralin-6-ol
MOL003283 CHEK1 (2R,3R,4S)-4-(4-hydroxy-3-methoxy-phenyl)-7-methoxy-2,3-dimethylol-tetralin-6-ol
MOL003283 NCOA2 (2R,3R,4S)-4-(4-hydroxy-3-methoxy-phenyl)-7-methoxy-2,3-dimethylol-tetralin-6-ol
MOL003283 SCN5A (2R,3R,4S)-4-(4-hydroxy-3-methoxy-phenyl)-7-methoxy-2,3-dimethylol-tetralin-6-ol
MOL003283 CCNA2 (2R,3R,4S)-4-(4-hydroxy-3-methoxy-phenyl)-7-methoxy-2,3-dimethylol-tetralin-6-ol
MOL003283 PTGS1 (2R,3R,4S)-4-(4-hydroxy-3-methoxy-phenyl)-7-methoxy-2,3-dimethylol-tetralin-6-ol
MOL004443 PTGS1 Zhebeiresinol
MOL004443 SCN5A Zhebeiresinol
MOL004443 PTGS2 Zhebeiresinol
MOL004443 RXRA Zhebeiresinol
MOL004443 ADRB2 Zhebeiresinol
MOL004443 GABRA1 Zhebeiresinol
MOL005828 NOS2 nobiletin
MOL005828 PTGS1 nobiletin
MOL005828 KCNH2 nobiletin
MOL005828 ESR1 nobiletin
MOL005828 AR nobiletin
MOL005828 PPARG nobiletin
MOL005828 PTGS2 nobiletin
MOL005828 F7 nobiletin
MOL005828 ESR2 nobiletin
MOL005828 CHEK1 nobiletin
MOL005828 PRSS1 nobiletin
MOL005828 NCOA2 nobiletin
MOL005828 GSK3B nobiletin
MOL005828 SCN5A nobiletin
MOL005828 BCL2 nobiletin
MOL005828 BAX nobiletin
MOL005828 CASP9 nobiletin
MOL005828 MMP9 nobiletin
MOL005828 JUN nobiletin
MOL005828 TP63 nobiletin
MOL005828 MAPK8 nobiletin
MOL005828 TIMP1 nobiletin
MOL005828 PPARG nobiletin
MOL005828 CREB1 nobiletin
MOL005828 PLA2G4A nobiletin
MOL005828 CD163 nobiletin
MOL005828 EPHB2 nobiletin
MOL007415 KCNH2 [(2S)-2-[[(2S)-2-(benzoylamino)-3-phenylpropanoyl]amino]-3-phenylpropyl] acetate
MOL007415 PTGS2 [(2S)-2-[[(2S)-2-(benzoylamino)-3-phenylpropanoyl]amino]-3-phenylpropyl] acetate
MOL007415 PRSS1 [(2S)-2-[[(2S)-2-(benzoylamino)-3-phenylpropanoyl]amino]-3-phenylpropyl] acetate
MOL007535 PGR (5S,8S,9S,10R,13R,14S,17R)-17-[(1R,4R)-4-ethyl-1,5-dimethylhexyl]-10,13-dimethyl-2,4,5,7,8,9,11,12,14,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthrene-3,6-dione
MOL009386 KCNH2 3,3′-bis-(3,4-dihydro-4-hydroxy-6-methoxy)-2H-1-benzopyran
MOL009386 ESR1 3,3′-bis-(3,4-dihydro-4-hydroxy-6-methoxy)-2H-1-benzopyran
MOL009386 PTGS2 3,3′-bis-(3,4-dihydro-4-hydroxy-6-methoxy)-2H-1-benzopyran
MOL009386 ADRB2 3,3′-bis-(3,4-dihydro-4-hydroxy-6-methoxy)-2H-1-benzopyran
MOL009386 CCNA2 3,3′-bis-(3,4-dihydro-4-hydroxy-6-methoxy)-2H-1-benzopyran