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. 2020 Feb 18;10(2):166–183. doi: 10.34172/apb.2020.022

Table 3. Account of recent paradigm CDs for drug Delivery .

Type of Cyclodextrin Molecule and category Route of administration Formulation Comments Ref.
2-hydroxy-propy-β-cyclodextrins (HPbetaCDs) Itraconazole (Antifungal) Pulmonary Aerosol Rapid absorption across the pulmonary epithelium compared to NP formulation of drug 124
Polymeric β-CDs Ethionamide (Antitubercular) Pulmonary Nanoparticles Drug incorporated following green protocol better for pulmonary administration 125
HP- β-CD Prednisolone and Fludrocortisone acetate (Corticosteroid) Pulmonary Dry powder aerosol CD promote dissolution and helps in permeation across a Calu-3 cell monolayer 126
Poly- β-CD Ethionamide (antitubercular) Pulmonary/ entdotracheal/ Intranasal Nanoparticles Empty Poly- β-CD has intrinsic antitubercular activity 127
Ethylenediamine derivative of​ β-​CD Doxorubicin HCl (Anticancer) Hep-G2 cell line study Magnetic nanocomposites NIR light −responsive controlled and targeted release 128
sulfobutylether- β-CD Naringenin (antimicrobial Anticancer) Ocular sulfobutylether- β-​CD/chitosan NPs CD/CS provided sustained release and improved bioavailability 129
µ-CD and γ-CD Cyclosporin (Immunosupressant) Ocular Nanoparticles γ -CD concentration has effects on aggregation but decreases particle size, safe for once or twice day administration 130
HP- β-​CD Resveratrol (Antioxidant) -- Polyvinylpyrrolidone-loaded resveratrol electrospinning nanofibers Improved aqueous solubility of drug with sutained drug release 131
βCD or HPbCD Glibenclamide (Hypoglycemic) Oral poly(anhydride) NPs CDs allow higher payload in NPs with initial burst release followed by sustained drug release 132
βCD Hyaluronic acid (anti-wrinkle effects and moisturizing agent) Transdermal quaternized βCD -grafted chitosan NPs Quaternization of CD gives stable NPs, water retention capacity of hyaluronic acid is improved by crosslinking with polymer 133
HP- β-CD, Methyl- β-CD and Trimethyl-β-CD Temoporfin (Photosensitizer for treatment of squamous cell carcinoma) -- Drug-in-cyclodextrin-in-liposome (DCL) nanoconstructs. trimethyl-β-CD-based DCL retains almost all drug and shows stability 134
HP-β-CD Dolutegravir sodium (DTG) Nose to brain delivery CD-based NPs CD-based NPs provided higher drug loading and 2.54 folds greater permeability of DTG compared to free drug 135
HP-β-CD Efavirenz (Antiviral) Intranasal chitosan-grafted-HPβCD NPs Chitosan and CD based NPs provide Sustained release, high brain targeted delivery and 4.76 times greater permeability than plain drug solution through porcine nasal mucosa. 136
HP-β-CD Benznidazole (Antiparasitic) -- Quatsomes and liposomes of CD based nanofomulates shows better activity against Trypanosoma cruzi as compared to drug and its nanostructure lipid carries. It contributes to the solubility of drug in formulation. 137
β-CD Curcumin (antioxidant, analgesic, anti-inflammatory and antiseptic) -- βCD based nanosponge (CDNS) Curcumin loaded CDNS shows the selective toxicity against cancerous cells and free CDNSs showed no toxicity 138
β-CD Saporin (Cytotoxic protein) -- βCD modified Circular bivalent aptamers (cb-apt) Supramolecular ensemble exhibits high serum stability, molecular recognition ability and enhanced intracellular delivery efficiency. 139
β-CD Doxorubicin (anticancer) HER2- Cell line study HApt aptamer-functionalized pH-sensitive β-CD-capped doxorubicin (DOX)-loaded mesoporous silica nanoparticles βCD works as pH sensitive nanovalve for DOX release 140

CD, cyclodextrin.