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. 2020 Apr 20;27(1):575–584. doi: 10.1080/10717544.2020.1748762

Table 1.

Oral pharmacokinetic parameters of TaxolTM (commercial formulation), PTX-loaded CS-SA micelles, PTX-loaded LC-SA/CS-SA micelles plus LC, and PTX-loaded LC-SA/CS-SA micelles in rats.

Parameters Taxol™ PTX-loaded CS-SA PTX-loaded LC-SA/ CS-SA + LC PTX-loaded LC-SA/ CS-SA
AUC(0–t) (mg/L·h) 28.98 24.43 28.24 48.05
t1/2z 83.83 44.85 30.78 9.40
Tmax (h) 0.5 2 2 2
Cmax (mg/L) 2.22 2.01 1.94 4.51
CLz/F (L/h/kg) 0.19 0.39 0.44 0.53
Vz/F (L/kg) 23.36 25.09 19.53 7.17
Relative bioavailability (%) 84.30 97.45 165.80
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