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. 2020 Mar 4;15(2):220–236. doi: 10.1016/j.ajps.2020.02.004

Table 1.

Distribution of transporters in tissues.

Position Influx transporter type Efflux transporter type
Intestine PEPT; OATPs; OCTNs; OCT1; OCT2 MDR1; MRP1/2/3/4/5; BCRP
Liver OATP1B1; OATP1B3; OATP2B1; OCT1; OAT2 MDR1/2/3; MRP2/3/4; BCRP; BSEP
Kidney OCT2; OAT1; OAT3; OAT4; PEPT2; GLUTs MDR1; MRP2/4; OCTN1/2; MATE1/2; OCT4; OATP1A2
Blood-brain barrier GLUT1; OAT3; OATP2B1; OCTN2; OCT1/2/3 MDR1; MRP1/2/3/4/5; BCRP