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. Author manuscript; available in PMC: 2020 May 7.

Published in final edited form as: Commun Chem. 2019 Jul 3;2:77. doi: 10.1038/s42004-019-0172-x

Table 2.

Displacement of [³H]rosiglitazone by sulfonamide compounds with recombinant human mitoNEET

Compounds	IC₅₀ (μM) ±std error	clogP^a
Furosemide	29.26 ±0.97	1.90
1	1021.00 ±0.96	1.11
2a	81.43 ±0.92	2.33
2b	42.56 ±1.03	2.86
2c	54.26 ±0.92	3.39
2d	9.12 ±1.04	3.92
2e	19.82 ±0.90	4.45
2f	6.24 ±0.88	4.98
2k	31.16 ± 1.02	3.31
2l	20.79 ± 1.01	2.72
2n	8.82 ± 1.00	2.87
2p	12.38 ± 1.23	2.37
Arachidonic acid	2.93 ± 1.06	6.3

^a

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