Skip to main content

View full-text article in PMC

. Author manuscript; available in PMC: 2021 May 1.

Published in final edited form as: Adv Biol Regul. 2020 Mar 10;76:100719. doi: 10.1016/j.jbior.2020.100719

Table 1.

X_I(50) values of cPLA₂ and iPLA₂ inhibitors.

			cPLA₂		iPLA₂
No	Code	Structure	% Inh.	X_I(50)	% Inh.	X_I(50)
1	643029 (Div. Set V)		94	1.5 ± 1	99	0.05 ± 0.01
2	6353053 (ChemBridge)		98	0.05 ± 0.05	100	0.1 ± 0.1
3	6937786 (ChemBridge)		98	0.3 ± 0.1	100	0.020 ± 0.008
4	20192 (Div. Set V)		97	0.2 ± 0.2	100	0.040 ± 0.005
5	204262 (Div. Set V)		94	0.5 ± 0.2	84	0.10 ± 0.08
6	46492 (Div. Set V)		96	0.03 ± 0.02	100	0.020 ± 0.005