Table 2.
Physicochemical Properties in vivo.
P.O. (10 mg/kg) | I.V. (2 mg/kg) | |
---|---|---|
T1/2 (hr) | 2.09 ± 0.93 | 4.41 ± 3.01 |
Tmax (hr) | 0.67 ± 0.29 | – |
Cmax (ng/mL) | 2753 ± 15.3 | – |
AUC0-t (ng·hr/mL) | 6203 ± 248 | 1842 ± 363 |
AUC0-∞ (ng·hr/mL) | 6315 ± 273 | 1854 ± 366 |
Vz_F(L/kg) | 4.79 ± 2.17 | 6.44 ± 4.09 |
Cl_F (mL/min/kg) | 26.4 ± 1.14 | 18.5 ± 3.9 |
MRT (hr) | 1.82 ± 0.35 | 1.25 ± 0.30 |
Bioavailability 68.1%.