Table 3.
Predicted human cytochrome P450 promiscuity of the proposed drugs.
Model Name | Azithromycin | Chloroquine | Lopinavir | Oseltamivir | Remdesivir | Ribavirin |
---|---|---|---|---|---|---|
CYP2D6 substrate | No | Yes | No | No | No | No |
CYP3A4 substrate | Yes | Yes | Yes | No | Yes | No |
CYP1A2 inhibitior | No | No | No | No | No | No |
CYP2C19 inhibitior | No | No | Yes | No | No | No |
CYP2C9 inhibitior | No | No | Yes | No | No | No |
CYP2D6 inhibitior | No | Yes | No | No | No | No |
CYP3A4 inhibitior | No | No | Yes | No | No | No |