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. 2020 May 15:1–11. doi: 10.1080/07391102.2020.1765876

Table 3.

Predicted human cytochrome P450 promiscuity of the proposed drugs.

Model Name Azithromycin Chloroquine Lopinavir Oseltamivir Remdesivir Ribavirin
CYP2D6 substrate No Yes No No No No
CYP3A4 substrate Yes Yes Yes No Yes No
CYP1A2 inhibitior No No No No No No
CYP2C19 inhibitior No No Yes No No No
CYP2C9 inhibitior No No Yes No No No
CYP2D6 inhibitior No Yes No No No No
CYP3A4 inhibitior No No Yes No No No