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. 2020 Feb 7;11(5):869–876. doi: 10.1021/acsmedchemlett.9b00656

Table 2. Permeability Assay Dataa.

Entry Papp AP (×10 –5 cm/s) Papp BL (×10 –5 cm/s) ER (Papp BL/Papp AP)
(±)-cis-1 3.7 ± 1.2 0.84 ± 0.20 0.22
Diazepam 2.0 ± 0.2 1.4 ± 0.2 0.70
FD-4 0.69 ± 0.10 0.65 ± 0.12 0.93
a

Values are mean ± SEM of three independent experiments.