Table 2. Permeability Assay Dataa.
Entry | Papp AP (×10 –5 cm/s) | Papp BL (×10 –5 cm/s) | ER (Papp BL/Papp AP) |
---|---|---|---|
(±)-cis-1 | 3.7 ± 1.2 | 0.84 ± 0.20 | 0.22 |
Diazepam | 2.0 ± 0.2 | 1.4 ± 0.2 | 0.70 |
FD-4 | 0.69 ± 0.10 | 0.65 ± 0.12 | 0.93 |
Values are mean ± SEM of three independent experiments.