Table 1. Peptide Segments Involved in PPIs.
PPI | peptide sequence | KD (μM) |
---|---|---|
menin/MLL1a | R6WRFPARPGTTGGGGGGGRR25 | 0.08212 |
MTIP/MyoAa | N799IPSLLRVQAHIRKKMVAQ818 | 0.08513 |
β-catenin/axina | E467NPESILDEHVQRVM481 | 514 |
Rab6a/Rab6IP1a | D900DEKEQFLYHLLSFNAV916 | 2015 |
ERα/NR-2Aa | H687KILHRLLQDS697 | 2.516 |
KCTD11/Cullin3a | N49SGLSFEELYRNAYTMVLHK68 | 0.49717 |
β-adaptin/β-arr.a | D383DDIVFEDFARQRLKGMKDD402 | 2.118 |
Bcl-XL/Baka | G72QVGRQLAIIGDDINR87 | 0.34019 |
Bcl-XL/Baxa | K57KLSECLKRIGDELDS72 | 1319 |
MDM2/p53a | Q16ETFSDLWKLLP27 | 0.06020 |
MDM2/p53a | F19SDLWKLL26 | 0.8021 |
MDM2/p53a | F19SDLWKL25 | 15021 |
Peptides are fragments of the indicated protein.