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. 2020 Feb 20;11(5):1047–1053. doi: 10.1021/acsmedchemlett.9b00620

Table 1. Peptide Segments Involved in PPIs.

PPI peptide sequence KD (μM)
menin/MLL1a R6WRFPARPGTTGGGGGGGRR25 0.08212
MTIP/MyoAa N799IPSLLRVQAHIRKKMVAQ818 0.08513
β-catenin/axina E467NPESILDEHVQRVM481 514
Rab6a/Rab6IP1a D900DEKEQFLYHLLSFNAV916 2015
ERα/NR-2Aa H687KILHRLLQDS697 2.516
KCTD11/Cullin3a N49SGLSFEELYRNAYTMVLHK68 0.49717
β-adaptin/β-arr.a D383DDIVFEDFARQRLKGMKDD402 2.118
Bcl-XL/Baka G72QVGRQLAIIGDDINR87 0.34019
Bcl-XL/Baxa K57KLSECLKRIGDELDS72 1319
MDM2/p53a Q16ETFSDLWKLLP27 0.06020
MDM2/p53a F19SDLWKLL26 0.8021
MDM2/p53a F19SDLWKL25 15021
a

Peptides are fragments of the indicated protein.