Figure 4. Mon1-Ccz1 activation by Rab5 is conserved in metazoan cells.
(A) Schematic representing the architecture of yeast and metazoan Rab7-GEF-complexes. Yeast Mon1-Ccz1 consists of a heterodimer whereas metazoan GEF-complex is a heterotrimer with Bulli (in Drosophila) or RMC1 in mammalian cells as a third subunit. A dimer of metazoan Mon1-Ccz1 may exist as well. (B) Purification and prenylation of Drosophila Rab-GTPases. Rab5 and Rab7 were prenylated and complexed with REP and GDI, respectively. (C) Purification of Drosophila dimeric and trimeric Rab7-GEF-complexes from insect cells as used for GEF-assays. (D) Recruiter GEF-assay with Drosophila dimeric and trimeric (Bulli-)Mon1-Ccz1. The recruiter GEF-assay was performed as described in Figure 3 using Drosophila protein complexes and increasing amounts of either Mon1-Ccz1 (Dimer) or Bulli-Mon1-Ccz1 (Trimer). (E) Enzymatic parameters as measured in (D). Values were calculated of two independent experiments. Error bars represent standard deviation. (F) Recruiter GEF-assay with decreasing amounts of Rab5. The recruiter-assay was performed as described above with 12.5 nM Mon1-Ccz1 and Bulli-Mon1-Ccz1, respectively, and the indicated amounts of recruiter Rab5. (G) Rate constants as derived from (F) in dependence of concentration of Rab5. Error bars represent standard deviation. For details see Methods.