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. Author manuscript; available in PMC: 2020 May 21.
Published in final edited form as: AAPS J. 2019 Sep 3;21(6):103. doi: 10.1208/s12248-019-0373-3

Table I.

Ratio of pharmacokinetic parameters (IV rifampin phase/control phase)

Drug AUCRifAUCCon CL/FRifCL/FCon Vss/FRifVss/FCon MRTRifMRTCon t12,zRift12,zCon
Atorvastatin 7.7 0.14 0.056 0.44 0.39
Rosuvastatin (Whites) 3.6 0.27 0.082 0.30 0.63
Rosuvastatin (Asians) 3.2 0.30 0.103 0.33 0.59
Glyburide (noninduced) 2.2 0.45 0.32 0.71 0.77
Glyburide (induced) 2.2 0.45 0.43 0.96 0.91