Table 8.
LoxA single-point screen inhibition percentages. Compounds are listed relative to their percent potency towards LoxA, with the most potent listed first. Each reaction contained 10 μM of A.A. and 25 μM inhibitor.
| NCGC00164603 | 95% | 76% | 33% | 23% | 0% |
| NCGC00015802 | 90% | 69% | 50% | 80% | 16% |
| NCGC00186032 | 87% | 57% | 36% | 78% | 5% |
| NCGC00015424 | 87% | 76% | 63% | 74% | 21% |
| NCGC00015280 | 86% | 51% | 38% | 42% | 0% |
| NCGC00018102 | 86% | 65% | 25% | 96% | 0% |
| NCGC00015300 | 83% | 65% | 48% | 41% | 13% |
| NCGC00024928 | 82% | 73% | 39% | 79% | 8% |
| NCGC00092386 | 76% | 51% | 26% | 83% | 5% |
| NCGC00091250 | 69% | 57% | 23% | 37% | 5% |