TABLE 4.
Coupling efficiencies for ligands at various primate OTRs
OTR | Potency/Affinity Ratio −Log(Ca2+ IC50/Ki) |
||
---|---|---|---|
Pro8-OT | Leu8-OT | AVP | |
Human | 2.51 | 2.75 | 2.80 |
Macaque | 1.51 | 1.57 | 1.77 |
Marmoset | 2.85 | 3.00 | 3.38 |
Titi monkey | 2.39 | 2.95 | 2.60 |
Coupling efficiencies for ligands at various primate OTRs
OTR | Potency/Affinity Ratio −Log(Ca2+ IC50/Ki) |
||
---|---|---|---|
Pro8-OT | Leu8-OT | AVP | |
Human | 2.51 | 2.75 | 2.80 |
Macaque | 1.51 | 1.57 | 1.77 |
Marmoset | 2.85 | 3.00 | 3.38 |
Titi monkey | 2.39 | 2.95 | 2.60 |