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. Author manuscript; available in PMC: 2020 May 28.
Published in final edited form as: ACS Chem Biol. 2019 Nov 12;14(12):2737–2744. doi: 10.1021/acschembio.9b00663

Table 2.

IC50 (μM) of Raloxifene and the Most Effective Analogsa

FpL2-6 H11G11 Rg3GUS Rh2GUS
raloxifene 78 ± 9 100 ± 5 13 ± 2 13 ± 3
UNC7084 18 ± 3 16 ± 3 5 ± 1 7 ± 3
UNC7087 15 ± 1 16 ± 1 4 ± 1 2 ± 1
UNC7159 13 ± 1 14 ± 1 7 ± 2 3 ± 1
a

Data are presented in micromolar as the average of 3 biological replicates ± SEM.