Table III.
MICs of zabofloxacin, moxifloxacin, levofloxacin and ciprofloxacin for selected 7 clinical MRSA isolates with detected mutations in QRDRs.
Strain No. | MIC (μg/ml) | Detected Mutation in QRDRs | |||||
---|---|---|---|---|---|---|---|
ZABa | MOX | LEV | CIP | gyrA | parC | parE | |
S37 | 4 | 8 | 32 | 64 | S84Lb | S80Fc | P451Sd |
S30 | 2 | 8 | 16 | 64 | S84L | S80F | P451S |
S5 | 2 | 4 | 16 | 64 | S84L | S80F | P451S |
S3 | 2 | 8 | 32 | 64 | S84L | S80F | P451S |
S11 | 0.125 | 0.25 | 8 | 32 | S84L | None | P451S |
S38 | 0.25 | 0.25 | 8 | 16 | None | S80F | None |
S22 | 0.03 | 0.25 | 4 | 8 | None | S80F | None |
ZAB: zabofloxacin, MOX: moxifloxacin, LEV: levofloxacin and CIP: ciprofloxacin.
Serine → Leucine,
Serine → Phenylalanine,
Proline → Serine.