Table 3.
Number of β-AR cells in different studies using radioligand methods
NUMBER OF β-AR IN CELL. MHMBRANK FRACTION | RADIOLIGAND BINDING ASSAY |
---|---|
~2,000 binding sites per lymphocyte in HC | 3H-alprenolol (19) |
~8,000 sites per lymphocyte in young and 14,000 old HC | 3H-dihydro-alprenolol (20) |
801 ± 114 sites per lymphocyte in elderly, 680 ± 47 in young HC | 3H-dihydro-alprenolol (21) |
2,230 ± 482 membrane β-AR per lymphocyte in inactive persons, 1,743 ± 85 per lymphocyte in active persons | 125I-cyanopindolol (22) |
2,499 ± 1,140 in untrained individuals, 2,366 ± 765 in baseball players, 1,634 ± 1,380 in short-distance runners, 1,446 ± long distance runner HC | 125I-cyanopindolol (23) |