Table 2:
IC50 and Hill coefficient values of 18 identified inhibitors
Name | IC50 (μM) | Hill Slope |
---|---|---|
Pimozide | 42 ± 2 | 3.1 ± 0.4 |
Ebastine | 57 ± 12 | 1.5 ± 0.2 |
Rupintrivir | 68 ± 7 | 1.4 ± 0.2 |
Bepridil | 72 ± 3 | 2.9 ± 1.0 |
Sertaconazole | 76 ± 2 | 3.5 ± 0.2 |
Rimonabant | 85 ± 3 | 5.0 ± 0.4 |
Oxiconazole | 99 ± 6 | 3.8 ± 0.4 |
Itraconazole | 111 ± 35 | 1.6 ± 0.2 |
Tipranavir | 180 ± 20 | 1.4 ± 0.2 |
Nelfinavir | 234 ± 15 | 5.4 ± 1.0 |
Zopiclone | 349 ± 77 | 1.2 ± 0.2 |
Trihexyphenidyl | 370 ± 53 | 8.9 ± 6.4 |
Saquinavir | 411 ± 6 | 26.8 ± 2.6 |
Isavuconazole | 438 ± 11 | 5.2 ± 0.7 |
Lopinavir | 486 ± 2 | 29.9 ± 2.4 |
Clemastine | 497 ± 148 | 11.2 ± 7.3 |
Metixene | 635 ± 43 | 8.7 ± 5 |
Duloxetine | 3047 ± 634 | 0.93 ± 0.07 |