Table 2.
Physicochemical characteristics of each liposomal preparation
| E-lipo | E/Asx-lipo | E/D-lipo | E/D/Asx-lipo | |
|---|---|---|---|---|
| Theoritical Asx concentration in liposomes (µM) | — | 200 | — | 200 |
| EPC concentration in liposome (mM) | 200 | 200 | 180 | 180 |
| DOTAP concentration in liposome (mM) | — | — | 20 | 20 |
| Particle diameter(nm) | 130.3 ± 6.6 | 131.2 ± 7.0 | 75.1 ± 7.5 | 84.6 ± 21.1 |
| PDI | 0.209 ± 0.033 | 0.279 ± 0.021 | 0.230 ± 0.015 | 0.281 ± 0.086 |
| Zeta potential (mV) | –0.88 ± 0.64 | –0.39 ± 0.53 | 8.68 ± 0.98 | 8.95 ± 1.07 |
| Actual Asx concentration in liposomes (µM) | — | 197.1 ± 0.9 | — | 203.8 ± 3.7 |
PDI, polydispersity index. Data are expressed as mean ± SD (n = 5).