Table 2.
Potency of TMEM16A Inhibitors Generated by QPatch Assay
| Name | IC50s (μM) for independent experiments |
||||
|---|---|---|---|---|---|
| 1 | 2 | 3 | 4 | 5 | |
| Benzbromarone | 3.45 | 1.51 | 1.31 | 2.30 | 3.18 |
| 1PBC | 1.18 | 0.85 | 1.10 | 1.57 | — |
| Niflumic acid | 5.29 | 4.62 | 8.45 | 11.12 | 7.71 |
| Niclosamide | 1.62 | 1.43 | 1.05 | 2.09 | 1.81 |
| Ani9 | 0.067 | 0.054 | 0.078 | — | — |
| AMG compound | 0.428 | 0.510 | 0.258 | 0.443 | 0.470 |