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. 2020 Apr 17;18(3):134–147. doi: 10.1089/adt.2019.962

Table 2.

Potency of TMEM16A Inhibitors Generated by QPatch Assay

Name IC50s (μM) for independent experiments
1 2 3 4 5
Benzbromarone 3.45 1.51 1.31 2.30 3.18
1PBC 1.18 0.85 1.10 1.57
Niflumic acid 5.29 4.62 8.45 11.12 7.71
Niclosamide 1.62 1.43 1.05 2.09 1.81
Ani9 0.067 0.054 0.078
AMG compound 0.428 0.510 0.258 0.443 0.470