| QSAR | Quantitative structure–activity relationship |
| HSVR | Hierarchical support vector regression |
| ADME/Tox | Absorption, distribution, metabolism and excretion, and toxicity |
| BDDCS | Biopharmaceutics drug disposition classification system |
| SLC | Solute carrier |
| ABC | ATP-binding cassette |
| Caco-2 | Colorectal adenocarcinoma |
| MDCK | Madin–Darby canine kidney |
| PAMPA | Parallel artificial membrane permeability assay |
| SPIP | Single-pass intestinal perfusion |