Table 4.
Performance for pKa Range 5.4–9.4; Programs Sorted Alphabetically
| program | number handled | predicted excellently (ADa ≤ 0.1) | predicted well (0.1 < AD ≤ 0.5) | predicted poorly (1.0 < AD ≤ 2.0) | predicted awfully (AD > 2.0) | r25.4–9.4 | MADb |
|---|---|---|---|---|---|---|---|
| ACD/pKa DB | 116 | 25 | 51 | 9 | 4 | 0.574 | 0.504 |
| ADME Boxes | 115 | 33 | 60 | 8 | 5 | 0.682 | 0.452 |
| ADMET Predictor | 116 | 14 | 53 | 15 | 8 | 0.350 | 0.744 |
| Epik | 114 | 9 | 29 | 39 | 9 | 0.403 | 0.979 |
| Jaguar | 84 | 10 | 16 | 20 | 9 | 0.422 | 1.044 |
| Marvin | 116 | 10 | 35 | 35 | 8 | 0.374 | 0.961 |
| Pallas pKalc | 115 | 21 | 45 | 19 | 6 | 0.469 | 0.680 |
| Pipeline Pilot | 114 | 35 | 30 | 28 | 10 | 0.422 | 0.762 |
| SPARC | 108 | 7 | 30 | 27 | 10 | 0.479 | 0.876 |
AD: absolute deviation.
MAD: mean absolute deviation.