Table 1. AR-V7 Expression Inhibitory Activity Evaluation for 1 and 3–5.
IC50 (nM) |
||||
---|---|---|---|---|
3 | 4 | 5 | spliceostatin A (1) | |
AR-V7-GFP negative population | 3.3 | 202 | 187 | 0.6 |
IC50 (nM) |
||||
---|---|---|---|---|
3 | 4 | 5 | spliceostatin A (1) | |
AR-V7-GFP negative population | 3.3 | 202 | 187 | 0.6 |