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. Author manuscript; available in PMC: 2020 Jul 1.
Published in final edited form as: Bioorg Chem. 2020 May 15;100:103934. doi: 10.1016/j.bioorg.2020.103934

Table 3.

IC50 of P10 and P19 on a panel of HDAC.

Compounds HDAC1 HDAC2 HDAC3 HDAC4 HDAC5 HDAC6 HDAC7 HDAC8
P10 >50 45 >50 >50 43 26 >50 23
P19 >50 41 >50 >50 >50 17 >50 9.3
PCI-34051* 3.0 45 38 10 >50 18 - 0.024
*

Kleinschek, A., et al. (2016). “Potent and Selective Non-hydroxamate Histone Deacetylase 8 Inhibitors.” ChemMedChem 11 (23): 2598–2606.