Table 3.
HPLC analysis of radiolabeled metabolites of [18F]FNDP in mouse blood and brain and baboon blood
| Met-1, % | Met-2, % | Parent [18F]FNDP, % | |
|---|---|---|---|
| Mouse blood (10 min) | 11.2 ± 4.8 | 25.4 ± 7.2 | 63.4 ± 4.4 |
| Mouse blood (30 min) | 10.1 ± 0.9 | 39.8 ± 9.8 | 50.1 ± 10.5 |
| Mouse brain (10 min) | 0.8 ± 0.3 | Nondetectable | 99.2 ± 0.3 |
| Mouse brain (30 min) | 1.7 ± 0.3 | Nondetectable | 98.3 ± 0.3 |
| Baboon blood (10 min) | 7.2 ± 1.9 | 15.8 ± 2.4 | 77.0 ± 3.6 |
| Baboon blood (30 min) | 16.7 ± 6.5 | 36.9 ± 3.1 | 46.5 ± 6.4 |
| Baboon blood (60 min) | 22.2 ± 9.3 | 49.5 ± 7.7 | 28.3 ± 9.3 |
| Baboon blood (90 min) | 22.3 ± 8.0 | 56.0 ± 7.1 | 21.8 ± 7.0 |