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. Author manuscript; available in PMC: 2020 Jun 24.
Published in final edited form as: Angew Chem Int Ed Engl. 2016 Aug 17;55(38):11382–11386. doi: 10.1002/anie.201603928

Figure 2.

Figure 2

Unlike the impermeable sulfone analog 7 (grey circles), 16 (black diamonds) displaces the ATAD2 bromodomain construct in a cellular nanoBRET displacement assay. 16 does not displace full-length ATAD2 (crosses). (Error bars = SD).