Table 5.
Small Molecules Targeting Host Factors and Unknown Targets
Name | Chemical structure | IC50 | Targets | Ref |
---|---|---|---|---|
Chlorpromazine (25) |
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7.24 μM | clathrin-mediated endocytosis | 122 |
fluphenazine (26) |
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3.23 μM | clathrin-mediated endocytosis | 122 |
promethazine (27) |
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7.48 μM | clathrin-mediated endocytosis | 122 |
imatinib (28) |
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10 μM | Abl2 | 123, 124 |
dasatinib (29) |
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2.1-5.4 μM | Abl | 125 |
saracatinib (30) |
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2.4-5.1 μM | SFK signaling pathways | 126 |
emodin (31) |
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200 μM | - | 131 |
SSAA09E3 (32) |
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9.7 μM | - | 57 |
VE607 (33) |
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1.6 μM | - | 132 |