TABLE 4.
Potencies of TxID and [V11L,V16D]ArIB for nAChR subtypes expressed in X. laevis oocytes
| IC50 values (nM) | ||||||||
|---|---|---|---|---|---|---|---|---|
| α3β2 | α3β4 | α4β2 | α4β4 | α6/α3β2β3 | α6/α3β4 | α7 | α9α10 | |
| TxID | >10,000a | 12.5a | >10,000a | >10,000a | >10,000a | 94.1a | >10,000a | >10,000a |
| [V11L,V16D]ArIB | >10,000b | >10,000b | >10,000 b | >10,000 b | 828 b | >10,000 b | 1.09b | >10,000b |
Luo et al., 2012