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. Author manuscript; available in PMC: 2021 Jul 1.
Published in final edited form as: J Neurochem. 2020 Feb 11;154(2):158–176. doi: 10.1111/jnc.14966

TABLE 4.

Potencies of TxID and [V11L,V16D]ArIB for nAChR subtypes expressed in X. laevis oocytes

IC50 values (nM)

α3β2 α3β4 α4β2 α4β4 α6/α3β2β3 α6/α3β4 α7 α9α10
TxID >10,000a 12.5a >10,000a >10,000a >10,000a 94.1a >10,000a >10,000a
[V11L,V16D]ArIB >10,000b >10,000b >10,000 b >10,000 b 828 b >10,000 b 1.09b >10,000b
a

Luo et al., 2012