Official websites use .gov
A
.gov website belongs to an official
government organization in the United States.
Secure .gov websites use HTTPS
A lock (
) or https:// means you've safely
connected to the .gov website. Share sensitive
information only on official, secure websites.
Kinase activity was measured by Caliper assay.
LTA-IL6 assay. All compounds were tested in duplicate unless otherwise noted.
Liver microsomal stability and kinome selectivity assays were typically single determinations. Kinome selectivity screens were done at a single concentration of 1 μM.
