Table I.
Leading drug candidates by antiretroviral class
| Antiretroviral Class | Leading Drug Candidate | Route of Administration | Phase of Development | FDA Approval |
|---|---|---|---|---|
| Capsid Inhibitors | GS-6207 | Oral, subcutaneous injection | Ib | No |
| Maturation Inhibitor | GSK2838232 | Oral | II | No |
| Nucleoside Reverse Transcriptase Translocation Inhibitors | Islatravir | Oral, subdermal implant | II | No |
| Anti-CD4 Monoclonal Antibodies | Ibalizumab | Infusion every 2 weeks | IV | Yes |
| Fusion Inhibitors | Albuvirtide | Intravenous injection | III | No |
| Non-Nucleoside Reverse Transcriptase Inhibitors | Elsulfavirine | Oral | II | No |
| Attachment Inhibitors | Fostemsavir | Oral | III | No |