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. 2020 Jul 21;10:12067. doi: 10.1038/s41598-020-69008-9

Table 1.

Ki(app) values (M) for TIMP-3 inhibition of selected metalloproteinases.

MMP-1ΔC (1 nM) 1.86E−9 ± 1.31E−10
MMP-3ΔC (1 nM) 5.50E−10 ± 4.48E−11
MMP-13 (0.1 nM) < 0.5 nM
ADAMTS-4 (0.5 nM) 1.24E−10 ± 3.95E−11
ADAMTS-5 (0.5 nM) 1.91E−09 ± 3.54E−11
ADAM17 (1 nM) 3.61E−09 ± 8.92E−11

Ki(app) given as mean ± standard deviation (n = 3–4).