Table 2.
Compound | ∗Binding constant (Ksv, M−1) | ¥IC50 (μM) |
---|---|---|
EA | 4.28 ± 0.28 × 104 | 39.7 ± 8.6 |
Quercetin | 7.82 ± 0.54 × 102 | 61.3 ± 5.4 |
∗Binding constant derived from fluorescence binding measurements. ¥IC50 value determined from enzyme inhibition assay.