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. Author manuscript; available in PMC: 2021 Mar 2.
Published in final edited form as: Adv Pharmacol. 2020 Mar 2;88:193–232. doi: 10.1016/bs.apha.2020.02.002

Table 1.

mGlu receptor PAMs and NAMs used in alcohol-related experiments.

Receptor PAM NAM Selected References
Group I
 mGlu1 CPCCOEt Schroeder et al., 2005; Hodge et al., 2006; Lominac et al., 2006
JNJ16259685 Besheer et al., 2008; Cozzoli et al., 2014; Lum et al., 2014
 
 mGlu5 CDPPB Gass et al., 2014; Gass et al., 2017
MPEP McGeehan and Olive, 2003; Backstrom et al., 2004; McMillen et al., 2005; Hodge et al., 2006; Lominac et al., 2006; Besheer et al., 2008; Gupta et al., 2008; Schroeder et al., 2008; Lee et al., 2016
MTEP Cowen et al., 2005; Cowen et al., 2007; Adams et al., 2008; Adams et al., 2010; Cozzoli et al., 2014; Lee et al., 2018; Gobin and Schwendt, 2019
Group II
 mGlu2 AZD8529 Augier et al., 2016; Li et al., 2016; Sidhpura et al., 2010
BINA Windisch and Czachowski, 2018
JNJ-42153605 Ahnaou et al., 2015, 2016
AZD8418 Li et al., 2016
LY487379 Nikiforuk et al., 2010;
Group III
 mGlu7 AMN082 (agonist) Bahi, 2012; Kotlinska et al., 2019