Table 1.
mGlu receptor PAMs and NAMs used in alcohol-related experiments.
Receptor | PAM | NAM | Selected References |
---|---|---|---|
Group I | |||
mGlu1 | CPCCOEt | Schroeder et al., 2005; Hodge et al., 2006; Lominac et al., 2006 | |
JNJ16259685 | Besheer et al., 2008; Cozzoli et al., 2014; Lum et al., 2014 | ||
mGlu5 | CDPPB | Gass et al., 2014; Gass et al., 2017 | |
MPEP | McGeehan and Olive, 2003; Backstrom et al., 2004; McMillen et al., 2005; Hodge et al., 2006; Lominac et al., 2006; Besheer et al., 2008; Gupta et al., 2008; Schroeder et al., 2008; Lee et al., 2016 | ||
MTEP | Cowen et al., 2005; Cowen et al., 2007; Adams et al., 2008; Adams et al., 2010; Cozzoli et al., 2014; Lee et al., 2018; Gobin and Schwendt, 2019 | ||
Group II | |||
mGlu2 | AZD8529 | Augier et al., 2016; Li et al., 2016; Sidhpura et al., 2010 | |
BINA | Windisch and Czachowski, 2018 | ||
JNJ-42153605 | Ahnaou et al., 2015, 2016 | ||
AZD8418 | Li et al., 2016 | ||
LY487379 | Nikiforuk et al., 2010; | ||
Group III | |||
mGlu7 | AMN082 (agonist) | Bahi, 2012; Kotlinska et al., 2019 |