Table 1.
Commercially marketed pharmaceuticals formulated with cyclodextrins throughout the world.
| Type | Drug name | Trade name | Route of Administration | Country |
|---|---|---|---|---|
| α-Cyclodextrin | Cefotiam hexetil hydrochloride | Pansporin T | Oral | Japan |
| β-Cyclodextrin | Omeprazole | Omebeta | Oral | Europe |
| Benexate hydrochloride | Ulgut, Lonmiel | Oral | Japan | |
| Chlordiazepoxide | Transilium | Oral | Argentina | |
| Nimesulide | Nimedex | Oral | Europe | |
| Nicotine | Nicorette | Sublingual | Europe | |
| Sulfobutylether β-Cyclodextrin | Carfilzomib | Kyprolis | Intravenous | Europe, USA |
| Ziprasidone Maleate | Geodon, Zeldox | Intramuscular | Europe, USA | |
| Aripiprazole | Abilify | Intramuscular | USA, Japan | |
| Voriconazole | Vfend | Intravenous | Europe, USA | |
| 2-Hydroxypropyl β-Cyclodextrin | Itraconazole | Sporanox | Oral, Intravenous | Europe, USA |
| Methylated β-Cyclodextrin | 17β-Estradiol | Aerodiol | Nasal | Europe |
| 2-Hydroxypropyl γ-Cyclodextrin | Diclofenac sodium | Voltaren | Ocular | Europe |