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[Preprint]. 2020 Jul 27:2020.07.24.20161547. [Version 1] doi: 10.1101/2020.07.24.20161547

Table 1.

Commercially marketed pharmaceuticals formulated with cyclodextrins throughout the world.

Type Drug name Trade name Route of Administration Country
α-Cyclodextrin Cefotiam hexetil hydrochloride Pansporin T Oral Japan
β-Cyclodextrin Omeprazole Omebeta Oral Europe
Benexate hydrochloride Ulgut, Lonmiel Oral Japan
Chlordiazepoxide Transilium Oral Argentina
Nimesulide Nimedex Oral Europe
Nicotine Nicorette Sublingual Europe
Sulfobutylether β-Cyclodextrin Carfilzomib Kyprolis Intravenous Europe, USA
Ziprasidone Maleate Geodon, Zeldox Intramuscular Europe, USA
Aripiprazole Abilify Intramuscular USA, Japan
Voriconazole Vfend Intravenous Europe, USA
2-Hydroxypropyl β-Cyclodextrin Itraconazole Sporanox Oral, Intravenous Europe, USA
Methylated β-Cyclodextrin 17β-Estradiol Aerodiol Nasal Europe
2-Hydroxypropyl γ-Cyclodextrin Diclofenac sodium Voltaren Ocular Europe