Skip to main content
. 2020 Jul 16;23(8):101377. doi: 10.1016/j.isci.2020.101377

Scheme 1.

Scheme 1

Scope of Amide Suzuki-Miyaura Cross-Coupling

Conditions: amide (1.0 equiv), Ar-B(OH)2 (2.0 equiv), [Pd(IPr)(μ-Cl)Cl]2, 0.25 mol%, K2CO3 (3.0 equiv), H2O (5 equiv), toluene (1.0 M), 23°C, 12 h. aIsolated yields. b0.50 mol%. d[Pd(IPr∗)(μ-Cl)Cl]2, 0.25 mol%. See Transparent Methods for details.