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. Author manuscript; available in PMC: 2020 Sep 1.
Published in final edited form as: J Clin Pharmacol. 2019 Sep;59(Suppl 1):S56–S69. doi: 10.1002/jcph.1489

Table 1.

Full Names, Protein Names, and Gene Names of Membrane Transporters Discussed in This Article

Full Name Protein Name Gene Name
P-glycoprotein P-gP ABCB1
Breast cancer resistance protein BCRP A8CG2
Multidrug and toxin extrusion 1 MATE 1 SLC47A1
Multidrug and toxin extrusion 2-K MATE2-K SLC47A2
Organic anion transporting polypeptide 1A2 OATP1A2 SLCO1A2
Organic anion transporting polypeptide 1B1 OATP1B1 SLCO1B1
Organic anion transporting polypeptide 1B3 OATP1B3 SLCO1B3
Organic anion transporting polypeptide 2B1 OATP2B1 SLCO2B1
Organic anion transporter 1 OAT1 SLC22A6
Organic anion transporter 3 OAT3 SLC22A8
Organic cation transporter 1 OCT1 SLC22A1
Organic cation transporter 2 OCT2 SLC22A2
Multidrug resistance-associated protein 1 MPR1 ABCC1
Multidrug resistance-associated protein 2 MRP2 ABCC2
Multidrug resistance-associated protein 3 MRP3 ABCC3
Multidrug resistance-associated protein 4 MRP4 ABCC4
Multidrug resistance-associated protein 6 MRP6 ABCC6
Peptide transporter 1 PEPT1 SLCI5A1
Sodium/taurocholate cotransporting polypeptide NTCP SLCIOA1
Bile salt export pump BSEP ABCB11
Glucose transporter 1 GLUTI SLC2A1
Glucose transporter 2 GLUT2 SLC2A2
Monocarboxylate transporter 1 MCT1 SLCI6A1
Uric acid transporter 1 URAT1 SLC22A12